Boron in drug discovery: carboranes as unique pharmacophores in biologically active compounds F Issa, M Kassiou, LM Rendina Chemical reviews 111 (9), 5701-5722, 2011 | 669 | 2011 |
Small animal SPECT and its place in the matrix of molecular imaging technologies SR Meikle, P Kench, M Kassiou, RB Banati Physics in Medicine & Biology 50 (22), R45, 2005 | 415 | 2005 |
DPA-714, a new translocator protein–specific ligand: Synthesis, radiofluorination, and pharmacologic characterization ML James, RR Fulton, J Vercoullie, DJ Henderson, L Garreau, S Chalon, ... Journal of Nuclear Medicine 49 (5), 814-822, 2008 | 294 | 2008 |
Molecular imaging of microglial activation in amyotrophic lateral sclerosis P Corcia, C Tauber, J Vercoullie, N Arlicot, C Prunier, J Praline, G Nicolas, ... PloS one 7 (12), e52941, 2012 | 280 | 2012 |
Low intrinsic efficacy for G protein activation can explain the improved side effect profiles of new opioid agonists A Gillis, AB Gondin, A Kliewer, J Sanchez, HD Lim, C Alamein, ... Science signaling 13 (625), eaaz3140, 2020 | 276 | 2020 |
Comparative evaluation of the translocator protein radioligands 11C-DPA-713, 18F-DPA-714, and 11C-PK11195 in a rat model of acute neuroinflammation F Chauveau, N Van Camp, F Dollé, B Kuhnast, F Hinnen, A Damont, ... Journal of Nuclear Medicine 50 (3), 468-476, 2009 | 265 | 2009 |
Neuroinflammation and brain atrophy in former NFL players: an in vivo multimodal imaging pilot study JM Coughlin, Y Wang, CA Munro, S Ma, C Yue, S Chen, R Airan, PK Kim, ... Neurobiology of disease 74, 58-65, 2015 | 261 | 2015 |
Pharmacology of Valinate and tert-Leucinate Synthetic Cannabinoids 5F-AMBICA, 5F-AMB, 5F-ADB, AMB-FUBINACA, MDMB-FUBINACA, MDMB-CHMICA, and … SD Banister, M Longworth, R Kevin, S Sachdev, M Santiago, J Stuart, ... ACS Chemical Neuroscience 7 (9), 1241-1254, 2016 | 259 | 2016 |
Pharmacology of indole and indazole synthetic cannabinoid designer drugs ab-fubinaca, adb-fubinaca, ab-pinaca, adb-pinaca, 5f-ab-pinaca, 5f-adb-pinaca, adbica, and 5f-adbica SD Banister, M Moir, J Stuart, RC Kevin, KE Wood, M Longworth, ... ACS chemical neuroscience 6 (9), 1546-1559, 2015 | 242 | 2015 |
Brain inflammation is induced by co-morbidities and risk factors for stroke C Drake, H Boutin, MS Jones, A Denes, BW McColl, JR Selvarajah, ... Brain, behavior, and immunity 25 (6), 1113-1122, 2011 | 241 | 2011 |
Recent developments in TSPO PET imaging as a biomarker of neuroinflammation in neurodegenerative disorders EL Werry, FM Bright, O Piguet, LM Ittner, GM Halliday, JR Hodges, ... International journal of molecular sciences 20 (13), 3161, 2019 | 237 | 2019 |
Effects of bioisosteric fluorine in synthetic cannabinoid designer drugs JWH-018, AM-2201, UR-144, XLR-11, PB-22, 5F-PB-22, APICA, and STS-135 SD Banister, J Stuart, RC Kevin, A Edington, M Longworth, SM Wilkinson, ... ACS Chemical Neuroscience 6 (8), 1445-1458, 2015 | 221 | 2015 |
Neuroinflammation in frontotemporal dementia F Bright, EL Werry, C Dobson-Stone, O Piguet, LM Ittner, GM Halliday, ... Nature Reviews Neurology 15 (9), 540-555, 2019 | 215 | 2019 |
Translational evaluation of translocator protein as a marker of neuroinflammation in schizophrenia T Notter, JM Coughlin, T Gschwind, U Weber-Stadlbauer, Y Wang, ... Molecular psychiatry 23 (2), 323-334, 2018 | 208 | 2018 |
Evaluation of the PBR/TSPO Radioligand [18F]DPA-714 in a Rat Model of Focal Cerebral Ischemia A Martín, R Boisgard, B Thézé, N Van Camp, B Kuhnast, A Damont, ... Journal of Cerebral Blood Flow & Metabolism 30 (1), 230-241, 2010 | 201 | 2010 |
The translocator protein AM Scarf, M Kassiou Journal of Nuclear Medicine 52 (5), 677-680, 2011 | 199 | 2011 |
An overview of late-stage functionalization in today’s drug discovery M Moir, JJ Danon, TA Reekie, M Kassiou Expert Opinion on Drug Discovery 14 (11), 1137-1149, 2019 | 185 | 2019 |
11C-DPA-713: a novel peripheral benzodiazepine receptor PET ligand for in vivo imaging of neuroinflammation H Boutin, F Chauveau, C Thominiaux, MC Grégoire, ML James, ... Journal of Nuclear Medicine 48 (4), 573-581, 2007 | 180 | 2007 |
Developing a preclinical model of Parkinson's disease: a study of behaviour in rats with graded 6-OHDA lesions L Truong, H Allbutt, M Kassiou, JM Henderson Behavioural brain research 169 (1), 1-9, 2006 | 174 | 2006 |
Imaging of glial cell activation and white matter integrity in brains of active and recently retired national football league players JM Coughlin, Y Wang, I Minn, N Bienko, EB Ambinder, X Xu, ME Peters, ... JAMA neurology 74 (1), 67-74, 2017 | 171 | 2017 |