Structure–activity relationships of benzimidazole derivatives as antiparasitic agents: dual activity-difference (DAD) maps J Pérez-Villanueva, R Santos, A Hernández-Campos, MA Giulianotti, ... MedChemComm 2 (1), 44-49, 2011 | 99 | 2011 |
Towards a systematic characterization of the antiprotozoal activity landscape of benzimidazole derivatives J Pérez-Villanueva, R Santos, A Hernández-Campos, MA Giulianotti, ... Bioorganic & medicinal chemistry 18 (21), 7380-7391, 2010 | 76 | 2010 |
Synthesis and antiprotozoal activity of novel 2-{[2-(1H-imidazol-1-yl) ethyl] sulfanyl}-1H-benzimidazole derivatives J Pérez-Villanueva, A Hernández-Campos, L Yépez-Mulia, ... Bioorganic & medicinal chemistry letters 23 (14), 4221-4224, 2013 | 70 | 2013 |
In vitro and in vivo trypanocidal activity of some benzimidazole derivatives against two strains of Trypanosoma cruzi DL Díaz-Chiguer, A Márquez-Navarro, B Nogueda-Torres, ... Acta tropica, 2012 | 59 | 2012 |
Synthesis and Biological Evaluation of 2H-Indazole Derivatives: Towards Antimicrobial and Anti-Inflammatory Dual Agents J Pérez-Villanueva, L Yépez-Mulia, I González-Sánchez, ... Molecules 22 (11), 1864, 2017 | 55 | 2017 |
Multitarget structure–activity relationships characterized by activity-difference maps and consensus similarity measure JL Medina-Franco, AB Yongye, J Pérez-Villanueva, RA Houghten, ... Journal of chemical information and modeling 51 (9), 2427-2439, 2011 | 54 | 2011 |
Antiprotozoal activity of proton-pump inhibitors J Pérez-Villanueva, A Romo-Mancillas, A Hernández-Campos, ... Bioorganic & medicinal chemistry letters 21 (24), 7351-7354, 2011 | 50 | 2011 |
Synthesis and in vitro cysticidal activity of new benzimidazole derivatives F Palomares-Alonso, H Jung-Cook, J Pérez-Villanueva, JC Piliado, ... European journal of medicinal chemistry 44 (4), 1794-1800, 2009 | 46 | 2009 |
Identifying Activity Cliff Generators of PPAR Ligands Using SAS Maps O Méndez‐Lucio, J Pérez‐Villanueva, R Castillo, JL Medina‐Franco Molecular Informatics, 2012 | 40 | 2012 |
Synthesis of curcuminoids and evaluation of their cytotoxic and antioxidant properties MC Lozada-García, RG Enríquez, TO Ramírez-Apán, A Nieto-Camacho, ... Molecules 22 (4), 633, 2017 | 38 | 2017 |
Activity cliffs and activity cliff generators based on chemotype-related activity landscapes J Pérez-Villanueva, O Méndez-Lucio, O Soria-Arteche, JL Medina-Franco Molecular diversity 19, 1021-1035, 2015 | 29 | 2015 |
Comparative molecular field analysis (CoMFA) and comparative molecular similarity indices analysis (CoMSIA) of some benzimidazole derivatives with trichomonicidal activity J Pérez-Villanueva, JL Medina-Franco, TR Caulfield, ... European journal of medicinal chemistry 46 (8), 3499-3508, 2011 | 29 | 2011 |
Casiopeinas of third generations: synthesis, characterization, cytotoxic activity and structure–activity relationships of mixed chelate compounds with bioactive secondary ligands Y Figueroa-DePaz, J Pérez-Villanueva, O Soria-Arteche, ... Molecules 27 (11), 3504, 2022 | 22 | 2022 |
Benzoic Acid Derivatives with Trypanocidal Activity: Enzymatic Analysis and Molecular Docking Studies toward Trans-Sialidase M Kashif, A Moreno-Herrera, JC Villalobos-Rocha, B Nogueda-Torres, ... Molecules 22 (11), 1863, 2017 | 20 | 2017 |
Activity landscape modeling of PPAR ligands with dual-activity difference maps O Méndez-Lucio, J Pérez-Villanueva, R Castillo, JL Medina-Franco Bioorganic & medicinal chemistry 20 (11), 3523-3532, 2012 | 20 | 2012 |
Indole-and pyrazole-glycyrrhetinic acid derivatives as PTP1B inhibitors: Synthesis, in vitro and in silico studies L De-la-Cruz-Martínez, C Duran-Becerra, M González-Andrade, ... Molecules 26 (14), 4375, 2021 | 17 | 2021 |
Synthesis, Antiprotozoal Activity, and Cheminformatic Analysis of 2-Phenyl-2H-Indazole Derivatives K Rodríguez-Villar, L Yépez-Mulia, M Cortés-Gines, JD Aguilera-Perdomo, ... Molecules 26 (8), 2145, 2021 | 17 | 2021 |
Chemoinformatic characterization of activity and selectivity switches of antiprotozoal compounds R Aguayo-Ortiz, J Pérez-Villanueva, A Hernández-Campos, R Castillo, ... Future Medicinal Chemistry 6 (3), 281-294, 2014 | 16 | 2014 |
CASE Plots for the Chemotype‐Based Activity and Selectivity Analysis: A CASE Study of Cyclooxygenase Inhibitors J Pérez‐Villanueva, JL Medina‐Franco, O Méndez‐Lucio, J Yoo, ... Chemical Biology & Drug Design 80 (5), 752-762, 2012 | 15 | 2012 |
3D-QSAR studies on purine-carbonitriles as cruzain inhibitors: comparative molecular field analysis (CoMFA) and comparative molecular similarity indices analysis (CoMSIA) O Méndez-Lucio, J Pérez-Villanueva, A Romo-Mancillas, R Castillo MedChemComm 2 (11), 1058-1065, 2011 | 15 | 2011 |