Chiral Oxazolopiperidone Lactams: Versatile Intermediates for the Enantioselective Synthesis of Piperidine‐Containing Natural Products C Escolano, M Amat, J Bosch Chemistry–A European Journal 12 (32), 8198-8207, 2006 | 243 | 2006 |
Enantioselective synthesis of piperidine, indolizidine, and quinolizidine alkaloids from a phenylglycinol-derived δ-lactam M Amat, N Llor, J Hidalgo, C Escolano, J Bosch The Journal of Organic Chemistry 68 (5), 1919-1928, 2003 | 207 | 2003 |
Synthesis of Enantiopure trans-3,4-Disubstituted Piperidines. An Enantiodivergent Synthesis of (+)- and (−)-Paroxetine M Amat, J Bosch, J Hidalgo, M Cantó, M Pérez, N Llor, E Molins, ... The Journal of Organic Chemistry 65 (10), 3074-3084, 2000 | 169 | 2000 |
Palladium (0)-catalyzed heteroarylation of 2-and 3-indolylzinc derivatives. An efficient general method for the preparation of (2-pyridyl) indoles and their application to … M Amat, S Hadida, G Pshenichnyi, J Bosch The Journal of Organic Chemistry 62 (10), 3158-3175, 1997 | 142 | 1997 |
A new synthetic entry to pentacyclic Strychnos alkaloids. Total synthesis of (.+-.)-tubifolidine,(.+-.)-tubifoline, and (.+-.)-19, 20-dihydroakuammicine M Amat, A Linares, J Bosch The Journal of Organic Chemistry 55 (26), 6299-6312, 1990 | 121 | 1990 |
Dynamic kinetic resolution of racemic γ-aryl-δ-oxoesters. Enantioselective synthesis of 3-arylpiperidines M Amat, M Cantó, N Llor, C Escolano, E Molins, E Espinosa, J Bosch The Journal of Organic Chemistry 67 (15), 5343-5351, 2002 | 97 | 2002 |
Enantioselective synthesis of 3, 3-disubstituted piperidine derivatives by enolate dialkylation of phenylglycinol-derived oxazolopiperidone lactams M Amat, O Lozano, C Escolano, E Molins, J Bosch The Journal of Organic Chemistry 72 (12), 4431-4439, 2007 | 95 | 2007 |
Preparation and reactions of 1-(tert-butyldimethylsilyl)-3-lithioindole. Regioselective synthesis of 3-substituted indoles M Amat, S Hadida, S Sathyanarayana, J Bosch The Journal of Organic Chemistry 59 (1), 10-11, 1994 | 93 | 1994 |
Identification of new aminoacid amides containing the imidazo [2, 1-b] benzothiazol-2-ylphenyl moiety as inhibitors of tumorigenesis by oncogenic Met signaling A Furlan, F Colombo, A Kover, N Issaly, C Tintori, L Angeli, V Leroux, ... European journal of medicinal chemistry 47, 239-254, 2012 | 91 | 2012 |
Chiral precursors for the synthesis of enantiomerically pure piperidines. Total synthesis of (R)-(-)-coniine M Amat, N Llor, J Bosch Tetrahedron letters 35 (14), 2223-2226, 1994 | 87 | 1994 |
Conjugate Addition of Organocuprates to Chiral Bicyclic δ-Lactams. Enantioselective Synthesis of cis-3,4-Disubstituted and 3,4,5-Trisubstituted Piperidines M Amat, M Pérez, N Llor, J Bosch, E Lago, E Molins Organic Letters 3 (4), 611-614, 2001 | 84 | 2001 |
Conjugate additions to phenylglycinol-derived unsaturated δ-lactams. Enantioselective synthesis of uleine alkaloids M Amat, M Pérez, N Llor, C Escolano, FJ Luque, E Molins, J Bosch The Journal of Organic Chemistry 69 (25), 8681-8693, 2004 | 82 | 2004 |
Straightforward Methodology for the Enantioselective Synthesis of Benzo[a]- and Indolo[2,3-a]quinolizidines M Amat, MMM Santos, O Bassas, N Llor, C Escolano, A Gómez-Esqué, ... The Journal of Organic Chemistry 72 (14), 5193-5201, 2007 | 75 | 2007 |
Dynamic kinetic resolution and desymmetrization processes: A straightforward methodology for the enantioselective synthesis of piperidines M Amat, O Bassas, N Llor, M Cantó, M Pérez, E Molins, J Bosch Chemistry–A European Journal 12 (30), 7872-7881, 2006 | 72 | 2006 |
Dynamic Kinetic Resolution and Desymmetrization of Enantiotopic Groups by Cyclodehydration of Racemic or Prochiral δ‐Oxoesters with (R)‐Phenylglycinol … M Amat, M Cantó, N Llor, V Ponzo, M Pérez, J Bosch Angewandte Chemie 114 (2), 345-348, 2002 | 69 | 2002 |
A biomimetic enantioselective approach to the decahydroquinoline class of dendrobatid alkaloids M Amat, R Griera, R Fabregat, E Molins, J Bosch Angewandte Chemie International Edition 47 (18), 3348-3351, 2008 | 66 | 2008 |
Total syntheses of the Strychnos indole alkaloids (−)-tubifoline,(−)-tubifolidine, and (−)-19, 20-dihydroakuammicine M Amat, MD Coll, J Bosch, E Espinosa, E Molins Tetrahedron: Asymmetry 8 (6), 935-948, 1997 | 66 | 1997 |
The strychnos alkaloids J Bosch, J Bonjoch, M Amat The alkaloids: chemistry and pharmacology, 75-189, 1996 | 59 | 1996 |
Enantioselective formal synthesis of (+)-dihydrocorynantheine and (−)-dihydrocorynantheol M Amat, A Gómez-Esqué, C Escolano, MMM Santos, E Molins, J Bosch The Journal of Organic Chemistry 74 (3), 1205-1211, 2009 | 56 | 2009 |
Preparation of enantiopure 6-(3-indolyl)-2-piperidones and conjugate additions to a 3, 4-didehydro derivative M Amat, N Llor, J Bosch, X Solans Tetrahedron 53 (2), 719-730, 1997 | 56 | 1997 |