Modern approaches for asymmetric construction of carbon–fluorine quaternary stereogenic centers: synthetic challenges and pharmaceutical needs Y Zhu, J Han, J Wang, N Shibata, M Sodeoka, VA Soloshonok, ... Chemical reviews 118 (7), 3887-3964, 2018 | 566 | 2018 |
Fluorine‐containing drugs approved by the FDA in 2018 H Mei, J Han, S Fustero, M Medio‐Simon, DM Sedgwick, C Santi, ... Chemistry–A European Journal 25 (51), 11797-11819, 2019 | 438 | 2019 |
Chemical aspects of human and environmental overload with fluorine J Han, L Kiss, H Mei, AM Remete, M Ponikvar-Svet, DM Sedgwick, ... Chemical Reviews 121 (8), 4678-4742, 2021 | 294 | 2021 |
Chiral sulfoxides: advances in asymmetric synthesis and problems with the accurate determination of the stereochemical outcome J Han, VA Soloshonok, KD Klika, J Drabowicz, A Wzorek Chemical Society Reviews 47 (4), 1307-1350, 2018 | 242 | 2018 |
Next generation organofluorine containing blockbuster drugs J Han, AM Remete, LS Dobson, L Kiss, K Izawa, H Moriwaki, ... Journal of Fluorine Chemistry 239, 109639, 2020 | 229 | 2020 |
Applications of fluorine-containing amino acids for drug design H Mei, J Han, KD Klika, K Izawa, T Sato, NA Meanwell, VA Soloshonok European journal of medicinal chemistry 186, 111826, 2020 | 197 | 2020 |
Fluorine-containing drugs approved by the FDA in 2019 H Mei, AM Remete, Y Zou, H Moriwaki, S Fustero, L Kiss, VA Soloshonok, ... Chinese Chemical Letters 31 (9), 2401-2413, 2020 | 191 | 2020 |
Cu-Catalyzed Deoxygenative C2-Sulfonylation Reaction of Quinoline N-Oxides with Sodium Sulfinate B Du, P Qian, Y Wang, H Mei, J Han, Y Pan Organic letters 18 (16), 4144-4147, 2016 | 154 | 2016 |
Recent advances on the electrochemical difunctionalization of alkenes/alkynes H Mei, Z Yin, J Liu, H Sun, J Han Chinese Journal of Chemistry 37 (3), 292-301, 2019 | 152 | 2019 |
Ni-catalyzed deaminative cross-electrophile coupling of Katritzky salts with halides via C─ N bond activation S Ni, CX Li, Y Mao, J Han, Y Wang, H Yan, Y Pan Science Advances 5 (6), eaaw9516, 2019 | 143 | 2019 |
Merging photoredox and copper catalysis: enantioselective radical cyanoalkylation of styrenes W Sha, L Deng, S Ni, H Mei, J Han, Y Pan ACS Catalysis 8 (8), 7489-7494, 2018 | 129 | 2018 |
Ni-catalyzed reductive cross-coupling of amides with aryl iodide electrophiles via C–N bond activation S Ni, W Zhang, H Mei, J Han, Y Pan Organic letters 19 (10), 2536-2539, 2017 | 122 | 2017 |
The self-disproportionation of enantiomers (SDE): a menace or an opportunity? J Han, O Kitagawa, A Wzorek, KD Klika, VA Soloshonok Chemical Science 9 (7), 1718-1739, 2018 | 120 | 2018 |
Iron-Catalyzed Cross-Dehydrogenative Coupling Esterification of Unactive C(sp3)–H Bonds with Carboxylic Acids for the Synthesis of α-Acyloxy Ethers J Zhao, H Fang, W Zhou, J Han, Y Pan The Journal of Organic Chemistry 79 (9), 3847-3855, 2014 | 116 | 2014 |
Synthesis of Chiral Sulfonyl Lactones via Copper‐Catalyzed Asymmetric Radical Reaction of DABCO⋅(SO2) Y Wang, L Deng, J Zhou, X Wang, H Mei, J Han, Y Pan Advanced Synthesis & Catalysis 360 (6), 1060-1065, 2018 | 114 | 2018 |
Tailor‐made amino acids and fluorinated motifs as prominent traits in modern pharmaceuticals H Mei, J Han, S White, DJ Graham, K Izawa, T Sato, S Fustero, ... Chemistry–A European Journal 26 (50), 11349-11390, 2020 | 113 | 2020 |
Assembly of fluorinated quaternary stereogenic centers through catalytic enantioselective detrifluoroacetylative aldol reactions C Xie, L Wu, J Han, VA Soloshonok, Y Pan Angewandte Chemie 127 (20), 6117-6121, 2015 | 110 | 2015 |
Self-disproportionation of enantiomers via sublimation; new and truly green dimension in optical purification J Han, D J Nelson, A E Sorochinsky, V A Soloshonok Current Organic Synthesis 8 (2), 310-317, 2011 | 108 | 2011 |
Fluorine-containing drugs approved by the FDA in 2021 J He, Z Li, G Dhawan, W Zhang, AE Sorochinsky, G Butler, ... Chinese Chemical Letters 34 (1), 107578, 2023 | 107 | 2023 |
Fluorine-containing pharmaceuticals approved by the FDA in 2020: Synthesis and biological activity Y Yu, A Liu, G Dhawan, H Mei, W Zhang, K Izawa, VA Soloshonok, J Han Chinese Chemical Letters 32 (11), 3342-3354, 2021 | 103 | 2021 |